| 5H-[1, 2, 4] Oxadiazolo [5, 4-d][1, 5] benzothiazepines as anticonvulsant agents in DBA/2 mice G De Sarro, A Chimirri, A De Sarro, R Gitto, S Grasso, M Zappalà European journal of medicinal chemistry 30 (12), 925-929, 1995 | 140 | 1995 |
| Pharmacophore‐based discovery of small‐molecule inhibitors of protein–protein interactions between HIV‐1 integrase and cellular cofactor LEDGF/p75 L De Luca, ML Barreca, S Ferro, F Christ, N Iraci, R Gitto, AM Monforte, ... ChemMedChem 4 (8), 1311-1316, 2009 | 139 | 2009 |
| 1-Aryl-3,5-dihydro-4H-2,3-benzodiazepin-4-ones: Novel AMPA Receptor Antagonists A Chimirri, G De Sarro, A De Sarro, R Gitto, S Grasso, S Quartarone, ... Journal of medicinal chemistry 40 (8), 1258-1269, 1997 | 116 | 1997 |
| Discovery of a novel and highly potent noncompetitive AMPA receptor antagonist R Gitto, ML Barreca, L De Luca, G De Sarro, G Ferreri, S Quartarone, ... Journal of medicinal chemistry 46 (1), 197-200, 2003 | 103 | 2003 |
| AMPA receptor antagonists as potential anticonvulsant drugs GD Sarro, R Gitto, E Russo, GF Ibbadu, ML Barreca, LD Luca, A Chimirri Current topics in medicinal chemistry 5 (1), 31-42, 2005 | 88 | 2005 |
| GYKI 52466 and related 2, 3-benzodiazepines as anticonvulsant agents in DBA/2 mice G De Sarro, A Chimirri, A De Sarro, R Gitto, S Grasso, P Giusti, ... European journal of pharmacology 294 (2-3), 411-422, 1995 | 85 | 1995 |
| Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor L De Luca, S Ferro, R Gitto, ML Barreca, S Agnello, F Christ, Z Debyser, ... Bioorganic & medicinal chemistry 18 (21), 7515-7521, 2010 | 80 | 2010 |
| Comparative anticonvulsant activity of some 2, 3-benzodiazepine derivatives in rodents G De Sarro, G Ferreri, P Gareri, E Russo, A De Sarro, R Gitto, A Chimirri Pharmacology Biochemistry and Behavior 74 (3), 595-602, 2003 | 78 | 2003 |
| Synthesis and anticonvulsant properties of 2, 3, 3a, 4-tetrahydro-1H-pyrrolo [1, 2-a] benzimidazol-1-one derivatives A Chimirri, A De Sarro, G De Sarro, R Gitto, M Zappala Il Farmaco 56 (11), 821-826, 2001 | 78 | 2001 |
| Synthesis and evaluation of pharmacological properties of novel annelated 2, 3-benzodiazepine derivatives R Gitto, V Orlando, S Quartarone, G De Sarro, A De Sarro, E Russo, ... Journal of medicinal chemistry 46 (17), 3758-3761, 2003 | 74 | 2003 |
| Exploiting the 1-(4-fluorobenzyl) piperazine fragment for the development of novel tyrosinase inhibitors as anti-melanogenic agents: Design, synthesis, structural insights and … L Ielo, B Deri, MP Germano, S Vittorio, S Mirabile, R Gitto, A Rapisarda, ... European journal of medicinal chemistry 178, 380-389, 2019 | 73 | 2019 |
| Synthesis and Evaluation of Pharmacological and Pharmacokinetic Properties of 11 H-[1, 2, 4] Triazolo [4, 5-c][2, 3] benzodiazepin-3 (2 H)-ones M Zappala, R Gitto, F Bevacqua, S Quartarone, A Chimirri, M Rizzo, ... Journal of medicinal chemistry 43 (25), 4834-4839, 2000 | 67 | 2000 |
| New AMPA antagonists in epilepsy E Russo, R Gitto, R Citraro, A Chimirri, G De Sarro Expert opinion on investigational drugs 21 (9), 1371-1389, 2012 | 66 | 2012 |
| Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as Potent Carbonic Anhydrase Inhibitors: Synthesis, Biological Evaluation, and Enzyme−Ligand X-ray … R Gitto, S Agnello, S Ferro, L De Luca, D Vullo, J Brynda, P Mader, ... Journal of medicinal chemistry 53 (6), 2401-2408, 2010 | 66 | 2010 |
| 3, 5-Dihydro-4 H-2, 3-benzodiazepine-4-thiones: a new class of AMPA receptor antagonists A Chimirri, G De Sarro, A De Sarro, R Gitto, S Quartarone, M Zappalà, ... Journal of medicinal chemistry 41 (18), 3409-3416, 1998 | 65 | 1998 |
| Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases L De Luca, F Mancuso, S Ferro, MR Buemi, A Angeli, S Del Prete, ... European journal of medicinal chemistry 143, 276-282, 2018 | 64 | 2018 |
| HIV-1 integrase strand-transfer inhibitors: design, synthesis and molecular modeling investigation L De Luca, S De Grazia, S Ferro, R Gitto, F Christ, Z Debyser, A Chimirri European journal of medicinal chemistry 46 (2), 756-764, 2011 | 64 | 2011 |
| Comparative anticonvulsant activity of N-acetyl-1-aryl-6, 7-dimethoxy-1, 2, 3, 4-tetrahydroisoquinoline derivatives in rodents G Ferreri, A Chimirri, E Russo, R Gitto, P Gareri, A De Sarro, G De Sarro Pharmacology Biochemistry and Behavior 77 (1), 85-94, 2004 | 57 | 2004 |
| Annelated 1, 5-benzodiazepines. I: Three, four, and five membered rings A Chimirri, R Gitto, S Grasso, AM Monforte, G Romeo, M Zappala Heterocycles (Sendai) 36 (3), 601-637, 1993 | 57 | 1993 |
| Structure-based screening for the discovery of new carbonic anhydrase VII inhibitors L De Luca, S Ferro, FM Damiano, CT Supuran, D Vullo, A Chimirri, R Gitto European Journal of Medicinal Chemistry 71, 105-111, 2014 | 55 | 2014 |
